Ark Pharm社　創薬研究用化合物

希少な化合物で創薬研究をサポート
創薬研究用化合物

Ark Pharm社は、創薬研究で役立つヘテロ環中間体、医薬品のビルディングブロックを取り扱っており、特にアルコール、アミン、アルデヒド、酸/エステル、ハロヘテロ環を含んだ化合物を数多く取り揃えています。今回は、他社で販売の少ない化合物の中から一部をご紹介します。

e-Nacalai Search Version の構造式検索では、構造式から簡便に弊社が取り扱う製品を一気に横断検索できます。また、簡易的な構造式作図ツールとしてもご活用いただけ、作図した構造式を他の構造式エディタでも開けるファイル形式で保存することも可能です。ぜひご活用ください。本サイトには、Ark Pharm社のみで登録されている製品が、約2000種類あります（2012年2月現在）。

特長

• 希少な化合物をラインアップ

製品紹介

ここでは、生理活性化合物の基本的な構成骨格とされているインドール骨格やインダゾール骨格をもつヘテロ環化合物の中から、一部を紹介します。

1-Boc-5-Chloro-6-trifluoromethyl-1H-indole	1'-Boc-1,2-dihydro-2-oxo-spiro[3H-indole-3,4'-piperidine]	1-Boc-3-Iodo-1H-indazole	5-Fluoro-1H-indazole-3-carboxylic Acid

■Ark Pharm社が取り揃えているヘテロ環構成骨格の種類

インドール、インダゾール、イミダゾール、ピラゾール、ピリダジン、ピリジン、ピリミジン、ピラジン、ピペラジン、ピペリジン、ピロリジン、チアゾール、トリアゾール

価格表

■ヘテロ環化合物

製品名	CAS No.	メーカー 製品番号	容量	価格	オンライン カタログへ
1-Boc-6-methyl-3-formylindole	914348-95-1	AK-16413	1 g	25,000
6-Benzyloxyindole-3-carbaldehyde	92855-64-6	AK-16427	1 g	25,000
5-Ethoxyindole	10501-17-4	AK-21810	1 g	30,000
5-Bromo-1H-indazole-3-carbaldehyde	201227-38-5	AK-22072	1 g	38,000
5-Methoxy-1H-indazole-3-carbaldehyde	169789-37-1	AK-22073	1 g	25,000
7-Methyl-1H-indazole-3-carbaldehyde	1000340-51-1	AK-22207	1 g	30,000
5-Fluoro-1H-indazole-3-carboxylic Acid	1077-96-9	AK-23992	1 g	45,000
1-Boc-5-chloro-6-trifluoromethyl-1H-indole	1209101-50-7	AK-24293	250 mg	45,000
1'-Boc-1,2-dihydro-2-oxo-spiro[3H-indole-3,4'-piperidine]	252882-60-3	AK-24410	250 mg	48,000
7-Fluoro-1H-indazole	341-24-2	AK-24464	1 g	18,000
5-Methoxy-7-azaindole	183208-36-8	AK-24543	250 mg	48,000
1-Boc-3-iodo-7-azaindole	192189-18-7	AK-24556	1 g	38,000
Methyl 4-Bromo-1H-indole-2-carboxylate	167479-13-2	AK-24952	250 mg	30,000
2-Methyl-7-azaindole	23612-48-8	AK-25051	250 mg	28,000
Methyl 3-Bromoindole-6-carboxylate	860457-92-7	AK-25193	1 g	23,000
N-Boc-1H-indole-6-carboxylic Acid Methyl Ester	957127-83-2	AK-25202	250 mg	25,000
3-Methyl-6-nitro-1H-indazole	6494-19-5	AK-26224	1 g	8,000
4-(1-Piperazinyl)-1H-indole	84807-09-0	AK-26360	250 mg	45,000
3-Bromo-5-nitroindazole	67400-25-3	AK-26734	1 g	5,000
6-Bromo-7-azaindole	143468-13-7	AK-27651	250 mg	48,000
3-Amino-5-nitroindazole	41339-17-7	AK-28420	1 g	15,000
4-Bromo-3-iodo-7-azaindole	1000340-34-0	AK-28632	250 mg	25,000
Ethyl 6-Chloroindole-2-carboxylate	27034-51-1	AK-29970	1 g	7,000
1-Boc-3-iodo-1H-indazole	290368-00-2	AK-31628	1 g	40,000
Ethyl 1-Methyl-7-oxo-4,5,6,7-tetrahydro-1H-indazole-3-carboxylate	802541-13-5	AK-32297	1 g	50,000
6-Trifluoromethyloxindole	1735-89-3	AK-33689	1 g	13,000
6-Bromo-1H-indazole-3-carbaldehyde	885271-72-7	AK-37707	250 mg	26,000
Methyl 6-Bromo-4-indolecarboxylate	107650-22-6	AK-39546	250 mg	48,000
5-Chloro-2-phenyl-1H-indole	23746-76-1	AK-45328	250 mg	32,000
2-Methyl-1-(4-nitrophenyl)-1H-imidazole	73225-15-7	AK-21719	1 g	15,000
1-(4-Nitrobenzyl)-1H-imidazole	18994-90-6	AK-21735	1 g	10,000
2-Methyl-1-(4-nitrobenzyl)-1H-imidazole	56643-86-8	AK-21741	1 g	13,000
3-Amino-6-bromopyrazine-2-carboxylic Acid	486424-37-7	AK-21914	1 g	20,000
Ethyl 1-Methyl-4-nitroimidazole-2-carboxylate	109012-23-9	AK-22184	1 g	18,000
2-n-Propyl-4-methyl-6-(1-methylbenzimidazole-2-yl)benzimidazole	152628-02-9	AK-23652	1 g	8,000
2-Amino-3-ethoxypyrazine	89464-86-8	AK-23934	250 mg	25,000
2-Amino-5-bromo-3-piperazin-1-ylpyrazine	893611-67-1	AK-23950	1 g	25,000
2-Amino-5-bromo-3-pyrrolidin-1-ylpyrazine	893611-72-8	AK-23951	1 g	25,000
2-Amino-5-bromo-3-(diethylamino)pyrazine	912773-09-2	AK-23955	1 g	25,000
2-Amino-5-bromo-6-chloropyrazine	173253-42-4	AK-23979	1 g	24,000
2-Amino-5-methoxypyrazine	54013-07-9	AK-24108	1 g	45,000
8-Chloroimidazo[1,2-a]pyrazine	69214-33-1	AK-24132	1 g	55,000
8-Chloro[1,2,4]triazolo[4,3-a]pyrazine	68774-77-6	AK-24563	1 g	50,000
N-Boc-2-amino-5-methylpyrazine	369638-68-6	AK-24726	1 g	38,000
2-Chloro-3-methoxypyrazine	40155-28-0	AK-25926	1 g	18,000
2-Amino-5-chloro-3-methoxypyrazine	874-31-7	AK-26837	250 mg	25,000
2-Chloro-6-methoxypyrazine	33332-30-8	AK-29172	1 g	11,000
Pyrazine-2-carbaldehyde	5780-66-5	AK-32007	1 g	45,000
5-Amino-1H-imidazole-4-carboxamide	21299-72-9	AK-34082	1 g	5,000
6-Bromo-3-iodoimidazo[1,2-a]pyrazine	1245644-42-1	AK-40672	1 g	40,000
2-[[[4-(3-Methoxypropoxy)-3-methylpyridine-2-yl]methyl]thio]-1H-benzimidazole	117977-21-6	AK-47315	1 g	15,000
2,6-Diaminopyrazine	41536-80-5	AK-50550	1 g	23,000

■フッ素化合物

製品名	CAS No.	メーカー 製品番号	容量	価格	オンライン カタログへ
2-(4-Fluorophenyl)thiazole-4-carboxylic Acid	863668-07-9	AK-22259	1 g	50,000
2-Fluoro-6-methylbenzoic Acid	90259-27-1	AK-23633	1 g	11,000
4-Ethyl-5-fluoropyrimidine	137234-88-9	AK-23771	1 g	8,000
2-Bromo-3'-trifluoromethoxyacetophenone	237386-01-5	AK-50568	1 g	15,000
1-Cyclopropyl-6-fluoro-7-chloro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic Acid	100361-18-0	AK-24774	1 g	20,000
2-Fluoro-3-methoxybenzoic Acid	137654-20-7	AK-24777	1 g	6,000
4-Cyano-2-fluorobenzaldehyde　劇	105942-10-7	AK-25279	1 g	11,000
2-Aminomethy-4-(4-fluorobenzyl)morpholine	112914-13-3	AK-25299	1 g	6,000
2-Cyclopropyl-4-(4-fluorophenyl)quinoline-3-carbaldehyde	121660-37-5	AK-25327	1 g	30,000
2[2-(4-Fluorophenyl)-2-oxo-1-phenylethyl]-4-methyl-3-oxo-pentanoic Acid Phenylamide	125971-96-2	AK-25339	1g	15,000
4-Bromo-3-fluorobenzonitrile　劇	133059-44-6	AK-25372	10 g	11,000
5-Chloro-2-fluorophenol	186589-76-4	AK-25539	1 g	18,000
4-Fluoro-3-nitrophenol	2105-96-6	AK-25593	1 g	20,000
2-Fluoro-3-nitrobenzoic Acid	317-46-4	AK-25758	1 g	8,000
2-Bromo-5-trifluoromethylphenol	402-05-1	AK-25928	1 g	5,000
3-Fluoro-4-nitroanisole	446-38-8	AK-25986	1 g	20,000
5-Bromo-2-(trifluoromethyl)aniline	703-91-3	AK-26279	1 g	13,000
1-Phenyl-5-trifluoromethyl-1H-pyrazole-4-carboxylic Acid Ethyl Ester	741717-63-5	AK-26306	250 mg	25,000
1-Bromo-3-fluoro-2-nitrobenzene	886762-70-5	AK-26408	1 g	9,000
3-Bromo-4-fluorophenol	27407-11-0	AK-26802	1 g	15,000
5'-Deoxy-5-fluorocytidine	66335-38-4	AK-26898	1 g	15,000
2-Fluoro-5-nitroanisole	454-16-0	AK-27026	1 g	5,000
2-Chloro-3-fluorobenzaldehyde	96516-31-3	AK-27086	1 g	16,000
2-Amino-4-fluorobenzonitrile　劇	80517-22-2	AK-27767	1 g	6,000
4-Fluoro-3-formylbenzonitrile　劇	146137-79-3	AK-28037	1 g	15,000
1-(5-Bromo-2-fluorophenyl)ethanone	198477-89-3	AK-28059	1 g	30,000
3-Bromo-2-fluorobenzadehyde	149947-15-9	AK-28788	1 g	4,000
2-Bromo-3-fluoro-6-picoline	374633-36-0	AK-29239	1 g	10,000
6-Fluoro-2-aminophenol	53981-25-2	AK-29356	1 g	30,000
2-Deoxy-2-fluoro-1,3,5-tri-O-benzoyl-alpha-D-arabinofuranose	97614-43-2	AK-29633	1 g	10,000
3-(Trifluoromethyl)-1H-pyrazole-4-carbaldehyde	1001020-14-9	AK-30440	250 mg	48,000

■光学活性化合物

製品名	CAS No.	メーカー 製品番号	容量	価格	オンライン カタログへ
(R)-N-Cbz-3,4-dihydro-1H-isoquinolinecarboxylic Acid	151004-88-5	AK-21839	250 mg	35,000
(S)-2-Methyl-1-(4-nitrobenzenesulfonyl)aziridine	374783-78-5	AK-21847	1 g	38,000
(R)-Azetidine-2-carboxylic Acid	7729-30-8	AK-23961	1 g	50,000
(S)-α,α-Diphenyl-3-pyrrolidineacetamide	133099-11-3	AK-24344	250 mg	35,000
(R)-2-Methylmorpholine	790184-33-7	AK-25482	250 mg	68,000
(R)-2-Aminopropanamide Hydrochloride	71810-97-4	AK-26287	1 g	8,000
(S)-2-Methylmorpholine	74572-13-7	AK-26310	250 mg	68,000
(S)-N-(2,6-Dimethylphenyl)-2-piperidinecarboxamide	27262-40-4	AK-27260	1 g	38,000
(R)-N-Boc-3-methylmorpholine	1022093-98-6	AK-28425	250 mg	86,000
(S)-N-Boc-3-methylmorpholine	1022094-01-4	AK-28426	250 mg	86,000
(S)-4-(4-Aminobenzyl)oxazolidin-2-one	340041-89-6	AK-28626	250 mg	40,000
(S)-3-Methylmorpholine	350595-57-2	AK-29208	1 g	70,000
(R)-1-Boc-2-benzylpiperazine	947684-78-8	AK-29661	250 mg	25,000
Methyl (R)-Piperidine-2-carboxylate	43041-11-8	AK-29738	1 g	38,000
(S)-(Piperidin-3-yl)methanol	144539-77-5	AK-29863	1 g	45,000
(R)-1-Boc-2-isopropylpiperazine	674792-04-2	AK-30116	1 g	50,000
(R)-1-Boc-2-ethylpiperazine	393781-70-9	AK-30321	1 g	40,000
(S)-3-Aminotetrahydrofuran Hydrochloride	204512-95-8	AK-32266	250 mg	25,000
(R)-3-Aminotetrahydrofuran Hydrochloride	1072015-52-1	AK-32944	250 mg	25,000
(R)-1-tert-Butyl 2-Methyl 5-Oxopyrrolidine-1,2-dicarboxylate	128811-48-3	AK-33083	1 g	16,000
(R)-1-(2,6-Dichloro-3-fluorophenyl)ethanol	330156-50-8	AK-34720	1 g	45,000
(R)-2-Aminocyclohenanol Hydrochloride	931-16-8	AK-36901	1 g	13,000
(S)-Methyl 2,3-Dihydroxypropanoate	10303-88-5	AK-39083	1 g	40,000
(R)-N-(2-Propynyl)-2,3-dihydroinden-1-amine	136236-51-6	AK-39976	1 g	30,000
(R)-1-Cbz-2-(aminomethyl)pyrrolidine	1187931-23-2	AK-40806	1 g	33,000
(S)-3-Methyl-1-(2-piperidinophenyl)butylamine N-Acetylglutamate	219921-94-5	AK-41426	1 g	8,000
(S)-(-)-3-(N-Methylamino)-1-(2-thienyl)-1-propanol	116539-55-0	AK-46639	1 g	10,000
(R)-3-(Cbz-amino)-5-oxotetrahydrofuran	118399-28-3	AK-47529	1 g	30,000
(R)-(-)-2-Phenylglycine Chloride Hydrochloride	39878-87-0	AK-48226	1 g	6,000
(S)-3-Hydroxybutyric Acid tert-Butyl Ester	82578-45-8	AK-49010	1 g	25,000

■ボロン酸

製品名	CAS No.	メーカー 製品番号	容量	価格	オンライン カタログへ
Benzylboronic Acid	4463-42-7	AK-23881	1 g	30,000
1-Boc-5,6-dichloro-1H-indole-2-boronic Acid	1310384-28-1	AK-24288	250 mg	65,000
1-Boc-6-fluoro-1H-indole-2-boronic Acid	1000068-26-7	AK-24289	250 mg	45,000
1-Tosyl-1H-pyrrolo[2,3-b]pyridin-3-ylboronic Acid	882562-39-2	AK-27364	250 mg	65,000
4'-Ethyl-4-biphenylboronic Acid	153035-62-2	AK-33429	1 g	13,000
3-(N,N-Dimethylamino)phenylboronic Acid Hydrochloride	1256355-23-3	AK-33777	1 g	6,000
N-Boc-1H-pyrazole-4-boronic Acid	947533-31-5	AK-39759	1 g	30,000
3,4,5-Trichlorophenylboronic Acid	862248-93-9	AK-44974	1 g	25,000
(3-Chloro-4-ethoxy-2-fluorophenyl)boronic Acid	909122-50-5	AK-49135	1 g	16,000

■カルボン酸

製品名	CAS No.	メーカー 製品番号	容量	価格	オンライン カタログへ
2-Aminothiazole-4-carboxylic Acid	40283-41-8	AK-15128	5 g	15,000
2-Amino-5-chlorothiazole-4-carboxylic Acid Methyl Ester	914348-76-8	AK-15130	1 g	16,000
3-(4-Chlorophenyl)piperazine-1-carboxylic Acid tert-Butyl Ester	886767-49-3	AK-16332	1 g	45,000
N-Cbz-2-piperidinecarboxylic Acid	71170-88-2	AK-17105	5 g	5,000
1-Pyridin-4-ylmethylpiperidine-4-carboxylic Acid	774531-43-0	AK-17129	1 g	18,000
4-(4-Aminophenyl)piperazine-1-carboxylic Acid tert-Butyl Ester	170911-92-9	AK-21754	1 g	15,000
3-Bromo-6-chloropyridine-2-carboxylic Acid	929000-66-8	AK-39554	1 g	23,000
5-Bromothiazole-4-carboxylic Acid	103878-58-6	AK-22047	1 g	30,000
2-(4-Methoxyphenyl)thiazole-4-carboxylic Acid	57677-80-2	AK-22271	1 g	50,000
2-Methylpyrimidine-4-carboxylic Acid	13627-49-1	AK-23648	1 g	45,000
4,6-Dimethylpyrimidine-5-carboxylic Acid	157335-93-8	AK-24036	1 g	19,000
1-(Phenoxycarbonyl)pyrrolidine-2-carboxylic Acid	1161602-22-7	AK-40068	1 g	38,000
5-Bromo-2-pyridinecarboxylic Acid Ethyl Ester	77199-09-8	AK-26326	1 g	30,000